{"id":55206,"date":"2024-01-11T14:36:31","date_gmt":"2024-01-11T14:36:31","guid":{"rendered":"https:\/\/medsname.com\/azopt-eye-drops\/"},"modified":"2026-04-30T10:24:50","modified_gmt":"2026-04-30T10:24:50","slug":"azopt-eye-drops","status":"publish","type":"product","link":"https:\/\/medsbase.com\/cs\/product\/azopt-eye-drops\/","title":{"rendered":"Azopt o\u010dn\u00ed kapky"},"content":{"rendered":"<p><!-- medsbase-tldr-answer --><\/p>\n<div class=\"medsbase-tldr-answer\" style=\"background:#fffbe6;border-left:4px solid #f5a623;padding:14px 18px;margin:14px 0 22px;border-radius:6px;font-size:15px;line-height:1.55;\">\n<h3 style=\"margin:0 0 6px;font-size:17px;color:#8a6d3b;\">\u26a1 Quick Answer \u2014 What is Azopt Eye Drops?<\/h3>\n<p style=\"margin:0;\">Azopt Eye Drops is Brinzolamide 1%, a carbonic anhydrase inhibitor (CAI) eye drop that lowers eye pressure 18\u201322% by reducing aqueous humour production. Used three times daily as monotherapy or twice daily as add-on. Avoid in severe sulfa allergy.<\/p>\n<\/div>\n<div class=\"medsbase-trust-strip\" style=\"background:#f6f7fb;border:1px solid #e3e5ee;border-radius:8px;padding:14px 18px;margin:18px 0;font-size:14px;line-height:1.55;\"><strong style=\"color:#1f3661;\">Pro\u010d objedn\u00e1vat z MedsBase?<\/strong> Dod\u00e1v\u00e1no od v\u00fdrobce certifikovan\u00e9ho WHO-GMP \u00b7 Diskr\u00e9tn\u00ed balen\u00ed \u00b7 Doprava po cel\u00e9m sv\u011bt\u011b \u00b7 <a href=\"\/cs\/reviews\/\" rel=\"noopener\">1 400+ ov\u011b\u0159en\u00fdch recenz\u00ed z\u00e1kazn\u00edk\u016f<\/a><\/div>\n<p class=\"medsbase-reship-line\" style=\"font-size:14px;color:#444;margin:8px 0 18px;\">\ud83d\udce6 Ka\u017ed\u00e1 objedn\u00e1vka je pokryta na\u0161\u00ed <a href=\"https:\/\/medsbase.com\/cs\/medsbase-re-shipment-assurance-policy\/\"><strong>Z\u00e1rukou op\u011btovn\u00e9ho odesl\u00e1n\u00ed<\/strong><\/a> \u2014 pokud va\u0161e z\u00e1silka nedoraz\u00ed do 20 pracovn\u00edch dn\u016f, p\u0159epos\u00edl\u00e1me ji.<\/p>\n<h3>Pro\u010d objedn\u00e1vat z MedsBase<\/h3>\n<p>Azopt Eye Drops is sourced from a WHO-GMP certified manufacturer and shipped worldwide in plain, discreet packaging. Every order is covered by our <a href=\"\/cs\/medsbase-re-shipment-assurance-policy\/\" rel=\"noopener\">Z\u00e1rukou op\u011btovn\u00e9ho odesl\u00e1n\u00ed<\/a> \u2014 pokud nedoraz\u00ed do 20 pracovn\u00edch dn\u016f, p\u0159epos\u00edl\u00e1me bez dal\u0161\u00edch n\u00e1klad\u016f. Podpo\u0159eno v\u00edce ne\u017e 1 400 ov\u011b\u0159en\u00fdmi recenzemi z\u00e1kazn\u00edk\u016f.<\/p>\n<h2>What is Azopt Eye Drops?<\/h2>\n<p>Azopt Eye Drops is manufactured by Alcon and contains Brinzolamide 1% as a sterile ophthalmic opaque suspension. It is a topical carbonic anhydrase inhibitor used to lower IOP in glaucoma. Brinzolamide is formulated as a milky-white suspension \u2014 shake well before each use. The suspension formulation has a near-neutral pH and tends to sting less than dorzolamide on instillation.<\/p>\n<h2>Jak to funguje<\/h2>\n<p>Brinzolamide blocks carbonic anhydrase isoenzyme II in the ciliary epithelium, slowing the formation of bicarbonate and the consequent flow of sodium and water into the posterior chamber. The result is reduced aqueous humour production and lower IOP. Topical CAIs reach significant intraocular concentration without the systemic side effects of oral acetazolamide (paraesthesia, kidney stones, taste disturbance).<\/p>\n<h2>Indikace &amp; D\u00e1vkov\u00e1n\u00ed<\/h2>\n<table style=\"width:100%;border-collapse:collapse;margin:14px 0;\">\n<thead>\n<tr style=\"background:#2c7cb0;color:#fff;\">\n<th style=\"padding:8px;text-align:left;border:1px solid #ddd;\">Indikace<\/th>\n<th style=\"padding:8px;text-align:left;border:1px solid #ddd;\">D\u00e1vka<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td style=\"padding:8px;border:1px solid #ddd;\">Monoterapie<\/td>\n<td style=\"padding:8px;border:1px solid #ddd;\">1 kapka do posti\u017een\u00e9ho oka t\u0159ikr\u00e1t denn\u011b<\/td>\n<\/tr>\n<tr style=\"background:#f9f9f9;\">\n<td style=\"padding:8px;border:1px solid #ddd;\">Dopl\u0148kov\u00e1 l\u00e9\u010dba k beta-blok\u00e1toru nebo PGA<\/td>\n<td style=\"padding:8px;border:1px solid #ddd;\">1 kapka dvakr\u00e1t denn\u011b<\/td>\n<\/tr>\n<tr>\n<td style=\"padding:8px;border:1px solid #ddd;\">Pokud suspenze<\/td>\n<td style=\"padding:8px;border:1px solid #ddd;\">Shake well before each instillation<\/td>\n<\/tr>\n<tr style=\"background:#f9f9f9;\">\n<td style=\"padding:8px;border:1px solid #ddd;\">V\u00edce kapek<\/td>\n<td style=\"padding:8px;border:1px solid #ddd;\">Po\u010dkejte 5 minut mezi r\u016fzn\u00fdmi p\u0159\u00edpravky<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<h2>Vedlej\u0161\u00ed \u00fa\u010dinky<\/h2>\n<p><strong>Lok\u00e1ln\u00ed:<\/strong> blurred vision (common with the suspension formulation \u2014 blink several times to clear), stinging on instillation (minimal), bitter taste in mouth (drainage through nasolacrimal duct), conjunctival hyperaemia, ocular pruritus, eyelid reactions.<\/p>\n<p><strong>Syst\u00e9mov\u00e9:<\/strong> bolest hlavy, \u00fanava (vz\u00e1cn\u00e9), ledvinov\u00e9 kameny (velmi vz\u00e1cn\u00e9 p\u0159i topick\u00e9m pou\u017eit\u00ed, na rozd\u00edl od peror\u00e1ln\u00edho acetazolamidu).<\/p>\n<div style=\"background:#fff3f3;border-left:4px solid #d9534f;padding:12px 16px;margin:14px 0;border-radius:4px;font-size:14px;line-height:1.55;\"><strong style=\"color:#a94442;\">Varov\u00e1n\u00ed p\u0159ed zk\u0159\u00ed\u017eenou reaktivitou se sulfonamidy.<\/strong> Jak brinzolamid, tak dorzolamid jsou deriv\u00e1ty sulfonamidu. U pacient\u016f se z\u00e1va\u017enou alergi\u00ed na sulfonamidy (Stevens-Johnson\u016fv syndrom, anafylaxe na sulfamethoxazol) se vz\u00e1cn\u011b vyvinuly zk\u0159\u00ed\u017een\u00e9 reakce. Anamn\u00e9za m\u00edrn\u00e9 vyr\u00e1\u017eky po sulfonamidech nen\u00ed absolutn\u00ed kontraindikac\u00ed, ale proberte to se sv\u00fdm l\u00e9ka\u0159em. V\u011bt\u0161ina reakc\u00ed je m\u00edrn\u00e9 konjunktiv\u00e1ln\u00ed podr\u00e1\u017ed\u011bn\u00ed sp\u00ed\u0161e ne\u017e syst\u00e9mov\u00e1 p\u0159ecitliv\u011blost.<\/div>\n<h2>Varov\u00e1n\u00ed a kontraindikace<\/h2>\n<ul>\n<li>T\u011b\u017ek\u00e1 p\u0159ecitliv\u011blost na sulfonamidy<\/li>\n<li>T\u011b\u017ek\u00e9 ren\u00e1ln\u00ed po\u0161kozen\u00ed (CrCl &lt; 30 ml\/min) \u2014 mo\u017en\u00e1 kumulace<\/li>\n<li>T\u011b\u017ek\u00e9 jatern\u00ed po\u0161kozen\u00ed<\/li>\n<li>Sou\u010dasn\u00e9 pod\u00e1v\u00e1n\u00ed peror\u00e1ln\u00edch inhibitor\u016f karboanhydr\u00e1zy (acetazolamid, methazolamid) \u2014 aditivn\u00ed \u00fa\u010dinek, ale omezen\u00fd dal\u0161\u00ed benefit<\/li>\n<li>Dysfunkce endotelu rohovky (Fuchsova dystrofie, stav po transplantaci rohovky) \u2014 inhibitory karboanhydr\u00e1zy mohou zhor\u0161it otok rohovky<\/li>\n<li>T\u011bhotensk\u00e1 kategorie C \u2014 vyvarujte se, pokud p\u0159\u00ednos nep\u0159ev\u00e1\u017e\u00ed riziko<\/li>\n<\/ul>\n<h2>Skladov\u00e1n\u00ed<\/h2>\n<p>Skladujte p\u0159i 15\u201325\u00b0C. Zlikvidujte 28 dn\u00ed po prvn\u00edm otev\u0159en\u00ed. Mezi pou\u017eit\u00edmi udr\u017eujte pevn\u011b uzav\u0159en\u00e9.<\/p>\n<h2 id=\"faqs\">\u010casto kladen\u00e9 dotazy<\/h2>\n<h3>What is the difference between Brinzolamide and acetazolamide?<\/h3>\n<p>Both target the same enzyme. Topical Brinzolamide delivers therapeutic levels at the eye with minimal systemic exposure. Oral acetazolamide produces systemic side effects (paraesthesia, taste changes, kidney stones, metabolic acidosis) that often limit long-term use.<\/p>\n<h3>Can I use Azopt Eye Drops if I&#039;m allergic to sulfa antibiotics?<\/h3>\n<p>Pokud jste m\u011bli Stevens-Johnson\u016fv syndrom nebo anafylaxi na sulfonamid, vyhn\u011bte se topick\u00fdm inhibitor\u016fm karboanhydr\u00e1zy. M\u00edrn\u00e1 vyr\u00e1\u017eka po sulfamethoxazolu nen\u00ed absolutn\u00ed kontraindikac\u00ed, ale p\u0159ed zah\u00e1jen\u00edm l\u00e9\u010dby se pora\u010fte se sv\u00fdm oftalmologem.<\/p>\n<h3>Why does Azopt Eye Drops make my mouth taste bitter?<\/h3>\n<p>After instillation, the drop drains through the nasolacrimal duct into the throat. Brinzolamide has a recognisable bitter taste. Punctal occlusion (pressing the inner corner of your eye for 1\u20132 minutes) reduces the effect.<\/p>\n<h3>How quickly does Azopt Eye Drops work?<\/h3>\n<p>Sn\u00ed\u017een\u00ed nitroo\u010dn\u00edho tlaku za\u010d\u00edn\u00e1 do 1 hodiny po prvn\u00ed d\u00e1vce; stabiln\u00ed \u00fa\u010dinek nast\u00e1v\u00e1 za 1\u20132 t\u00fddny. Pr\u016fm\u011brn\u00e9 sn\u00ed\u017een\u00ed je 18\u201322 % od v\u00fdchoz\u00ed hodnoty p\u0159i monoterapii.<\/p>\n<h3>Is the blurred vision after instilling Azopt Eye Drops normal?<\/h3>\n<p>Yes \u2014 brinzolamide is formulated as an opaque suspension, and a few minutes of mild blur after instillation is expected. Blink several times to clear. Avoid driving immediately after dosing.<\/p>\n<h3>Can I combine Azopt Eye Drops with other glaucoma drops?<\/h3>\n<p>Ano \u2014 inhibitory karboanhydr\u00e1zy (CAI) p\u016fsob\u00ed aditivn\u011b s beta-blok\u00e1tory, analogy prostaglandin\u016f a alfa-2 agonisty. Mezi aplikac\u00ed r\u016fzn\u00fdch lahvi\u010dek po\u010dkejte 5 minut. Pro lep\u0161\u00ed adherenci existuj\u00ed fixn\u00ed kombinace jako dorzolamid+timolol.<\/p>\n<h3>Co kdy\u017e zapomenu d\u00e1vku?<\/h3>\n<p>Vezm\u011bte si l\u00e9k, jakmile si vzpomenete, pokud nen\u00ed bl\u00edzko dal\u0161\u00ed napl\u00e1novan\u00e1 d\u00e1vka \u2014 v takov\u00e9m p\u0159\u00edpad\u011b vynechejte vynechanou d\u00e1vku. Ned\u00e1vejte dvojn\u00e1sobnou d\u00e1vku.<\/p>\n<h3>Can I use Azopt Eye Drops in pregnancy?<\/h3>\n<p>Kategorie C. Lok\u00e1ln\u00ed inhibitory karboanhydr\u00e1zy p\u0159estupuj\u00ed placentou v mal\u00e9m mno\u017estv\u00ed. Vyhn\u011bte se jim, pokud v\u00e1\u0161 oftalmolog nerozhodne, \u017ee p\u0159\u00ednos jasn\u011b p\u0159eva\u017euje riziko. Proberte alternativy jako brimonidin nebo selektivn\u00ed laserovou trabekuloplastiku.<\/p>\n<h3>Pro\u010d t\u0159ikr\u00e1t denn\u011b nam\u00edsto dvakr\u00e1t?<\/h3>\n<p>When used as monotherapy, Brinzolamide has an 8-hour duration so three-times-daily dosing maintains 24-hour IOP control. When added to an existing beta-blocker or prostaglandin, twice daily is sufficient because the partner drug provides additional coverage.<\/p>\n<h3>Co kdy\u017e mi z\u010derven\u00e1 nebo sv\u011bd\u00ed oko?<\/h3>\n<p>M\u00edrn\u00e9 zarudnut\u00ed spojivek je b\u011b\u017en\u00e9 v prvn\u00edch 1\u20132 t\u00fddnech a obvykle ustoup\u00ed. P\u0159etrv\u00e1vaj\u00edc\u00ed zarudnut\u00ed, otekl\u00e1 v\u00ed\u010dka nebo sv\u011bd\u011bn\u00ed mohou nazna\u010dovat hypersenzitivn\u00ed reakci \u2014 p\u0159esta\u0148te kapky pou\u017e\u00edvat a kontaktujte sv\u00e9ho oftalmologa.<\/p>\n<p><!-- medsbase-related-alts-v1 --><\/p>\n<h3>Dal\u0161\u00ed o\u010dn\u00ed l\u00e9ky<\/h3>\n<p>Z\u00e1kazn\u00edci, kte\u0159\u00ed si prohl\u00ed\u017eej\u00ed tento produkt, tak\u00e9 zva\u017euj\u00ed tyto alternativy v na\u0161\u00ed <a href=\"\/cs\/eye-care\/\">P\u00e9\u010de o o\u010di<\/a> nab\u00eddce:<\/p>\n<ul>\n<li><a href=\"https:\/\/medsbase.com\/cs\/xalatan-eye-drop\/\">Xalatan o\u010dn\u00ed kapky (latanoprost)<\/a><\/li>\n<li><a href=\"https:\/\/medsbase.com\/cs\/azopt-eye-drops\/\">Azopt o\u010dn\u00ed kapky (brinzolamid)<\/a><\/li>\n<li><a href=\"https:\/\/medsbase.com\/cs\/alphagan-p-drop\/\">Alphagan P kapky (brimonidin)<\/a><\/li>\n<li><a href=\"https:\/\/medsbase.com\/cs\/iotim-eye-drops\/\">Iotim o\u010dn\u00ed kapky (timolol)<\/a><\/li>\n<li><a href=\"https:\/\/medsbase.com\/cs\/careprost-eye-drops\/\">Careprost (bimatoprost)<\/a><\/li>\n<\/ul>\n<h3>L\u00e9ka\u0159sk\u00e9 upozorn\u011bn\u00ed<\/h3>\n<p style=\"font-size:13px;color:#555;\">Informace na t\u00e9to str\u00e1nce slou\u017e\u00ed pouze pro vzd\u011bl\u00e1vac\u00ed \u00fa\u010dely a nenahrazuj\u00ed l\u00e9ka\u0159skou pomoc kvalifikovan\u00e9ho oftalmologa nebo optometristy. O\u010dn\u00ed onemocn\u011bn\u00ed mohou rychle ohrozit zrak \u2014 n\u00e1hl\u00e1 ztr\u00e1ta zraku, siln\u00e1 bolest nebo trauma p\u0159edstavuj\u00ed oftalmologickou pohotovost. P\u0159ed zah\u00e1jen\u00edm, ukon\u010den\u00edm nebo zm\u011bnou jak\u00e9koli l\u00e9\u010dby se v\u017edy pora\u010fte s odborn\u00edkem na p\u00e9\u010di o zrak.<\/p>","protected":false},"excerpt":{"rendered":"<p>Azopt (brinzolamide 1%) \u2014 three-times-daily ophthalmic carbonic anhydrase inhibitor for open-angle glaucoma. Suspension \u2014 shake well. Sulfa cross-reactivity caution.<\/p>","protected":false},"featured_media":55207,"comment_status":"open","ping_status":"open","template":"","meta":[],"product_brand":[],"product_cat":[3141,3343,3342],"product_tag":[3876,3877],"class_list":{"0":"post-55206","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-category-overview","7":"product_cat-eye-care","8":"product_cat-general-health","9":"product_tag-azopt-eye-drops","10":"product_tag-brinzolamide","12":"first","13":"instock","14":"shipping-taxable","15":"purchasable","16":"product-type-variable","17":"has-default-attributes"},"acf":[],"_links":{"self":[{"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/product\/55206","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/comments?post=55206"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/media\/55207"}],"wp:attachment":[{"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/media?parent=55206"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/product_brand?post=55206"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/product_cat?post=55206"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/medsbase.com\/cs\/wp-json\/wp\/v2\/product_tag?post=55206"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}